Department Researches & Publications

Department of Medicinal Chemistry

Researches Our research spans a wide range from basic organic synthesis, drug design and development, structure elucidation of newly synthesized compound and natural products. The research focuses on the following strategic Research Themes: Design and synthesis of new chemical entities. Computer aided drug design studies. Structure-Activity relationship studies. Combinatorial chemistry. Prod rugs developments. Analytical methods for bioavailability and metabolic studies. Research within these Themes is carried out in multidisciplinary groupings focused on the discovery of novel techniques and/or enhancement of the already existing ones. At the department of Medicinal Pharmacy, We have major national and international collaborative research projects and a significant output of research publications in high-ranking journals. Our academic collaborators include many Universities in USA, Canada, Japan, and a number of major European universities.

# Title Research Year
121 Synthesis and In Vitro Evaluation of Ferutinol Aryl Esters for Estrogenic Activity and Affinity Toward Cannabinoid Receptors 2015
122 Synthesis, anti-inflammatory and molecular docking of some new 1,2,4-triazolobenzimidazol-3-yl acetone thiosemicarbazone cyclized derivatives as PLA-2 inhibitors 2015
123 Synthesis, Biological Investigation and Molecular Docking Study of N-Malonyl-1,2-dihydroisoquinoline Derivatives as Brain Specific and Shelf-Stable MAO Inhibitors 2015
124 Synthesis, Biological Investigation and Molecular Docking Study of N-Malonyl-1,2-dihydroisoquinoline Derivatives as Brain Specific and Shelf-Stable MAO Inhibitors 2015
125 Synthesis, Biological Investigation and Molecular Docking Study of N-Malonyl-1,2-dihydroisoquinoline Derivatives as Brain Specific and Shelf-Stable MAO Inhibitors 2015
126 Synthesis, Biological Investigation and Molecular Docking Study of N-Malonyl-1,2-dihydroisoquinoline Derivatives as Brain Specific and Shelf-Stable MAO Inhibitors 2015
127 Small-Molecule Inhibitors of 25-Hydroxyvitamin D-24-
Hydroxylase (CYP24A1): Synthesis and Biological Evaluation. 		2014
128 Charge-Transfer Reaction of 1,4-Benzoquinone with Crizotinib: Spectrophotometric Study, Computational Molecular Modeling and Use in Development of Microwell Assay for Crizotinib 2014
129 Design and synthesis of new pyrido[2,3-d]pyrimidine-1,4-dione derivatives as anti-inflammatory agents 2014
130 Development of quinone analogues as dynamin GTPase inhibitors 2014